Electron transfer induced deprotonation of α-and β-pinene: Evidence for ring-closed vinylcyclobutane radical cations

Dahui Zhou, Mohsin Sheik, Heinz D. Roth

Research output: Contribution to journalArticlepeer-review

14 Scopus citations

Abstract

Electron transfer from α-(1) or β-pinene (2), to 2,3,5,6-tetrachlorobenzoquinone generates radical cations, which are rapidly deprotonated by the semiquinone radical anion. (1S,5S)-2 is converted to (1S,5S)-1 and (1R,5R)-1 yields a dehydrogenation product, verbenene, (1R,5R)-9 with essentially quantitative retention of optical activity. The results support chiral, "ring-closed" radical cation structures in which the allylic-quaternary cyclobutane C-C bond retains a significant degree of bonding.

Original languageEnglish (US)
Pages (from-to)2385-2388
Number of pages4
JournalTetrahedron Letters
Volume37
Issue number14
DOIs
StatePublished - Apr 1 1996

All Science Journal Classification (ASJC) codes

  • Biochemistry
  • Drug Discovery
  • Organic Chemistry

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